3058600-77-1
Chemical Structure
Mu opioid receptor antagonist 9
- CAS No.: 3058600-77-1
- Formula:C21H27ClN2O2
- Molecular Weight:374.90
InChIKey: KOENSXNJMXLQDK-UHFFFAOYSA-N
SMILES: C=CCN(CCC1)CCCC1N(C(C2=COC=C2)=O)C3=CC=CC=C3.Cl
Biological Activity: Mu opioid receptor antagonist 9 is potent, selective and CNS-pentrant mu-opioid receptor (MOR) antagonist with a Ki of 77.3 nM. Mu opioid receptor antagonist 9 exhibits selectivity over kappa-opioid receptor (KOR), and delta-opioid receptor (DOR). Mu opioid receptor antagonist 9 effectively blocks the antinociceptive effects of psychoactive substances. Mu opioid receptor antagonist 9 can reverse psychoactive substances-induced respiratory depression in mice. Mu opioid receptor antagonist 9 can be used for the research of Opioid Use Disorder (OUD)[1].
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Mu opioid receptor antagonist 9 | Mu opioid receptor antagonist 9 is potent, selective and CNS-pentrant mu-opioid receptor (MOR) antagonist with a Ki of 77.3 nM. Mu opioid receptor antagonist 9 exhibits selectivity over kappa-opioid receptor (KOR), and delta-opioid receptor (DOR). Mu opioid receptor antagonist 9 effectively blocks the antinociceptive effects of psychoactive substances. Mu opioid receptor antagonist 9 can reverse psychoactive substances-induced respiratory depression in mice. Mu opioid receptor antagonist 9 can be used for the research of Opioid Use Disorder (OUD). | |||||||||||||||||||||
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