3086536-23-1
3086536-23-1
Chemical Structure
CDD-2807
- CAS No.: 3086536-23-1
- Formula:C29H26N4O
- Molecular Weight:446.54
InChIKey: YXMAOKMVGOSRPS-UHFFFAOYSA-N
SMILES: O=C(C1=CC2=C(NN=C2C#CC3=CC=CC=C3C4=CC=CC=C4)C=C1)N5CC6(CNCCC6)C5
Biological Activity: CDD-2807 is a blood-testis barrier-penetrant STK33 inhibitor (Kd = 0.02 nM). CDD-2807 acts by impairing sperm motility and hyperactivation, while inhibiting off-target kinases such as CLK4 (Kd = 0.9 nM), CLK2 (Ki = 1.3 nM), RET (Ki = 0.3 nM), and CLK1 (Ki = 3.1 nM). CDD-2807 can be used in research on reversible male contraception[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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CDD-2807 | 99.52% | CDD-2807 is a blood-testis barrier-penetrant STK33 inhibitor (Kd = 0.02 nM). CDD-2807 acts by impairing sperm motility and hyperactivation, while inhibiting off-target kinases such as CLK4 (Kd = 0.9 nM), CLK2 (Ki = 1.3 nM), RET (Ki = 0.3 nM), and CLK1 (Ki = 3.1 nM). CDD-2807 can be used in research on reversible male contraception. | ||||||||||||||||||||
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