3103571-04-3
3103571-04-3
Chemical Structure
GPR133 agonist 1
- CAS No.: 3103571-04-3
- Formula:C25H34N4O3
- Molecular Weight:438.56
InChIKey: WAEKNLBCKPEEKN-UHFFFAOYSA-N
SMILES: O=C(N(C)C)C1=CC=C(N2CCN(CC2)CC)C(NC(COC3=CC=C(C)C=C3C)=O)=C1
Biological Activity: GPR133 agonist 1 is an orally active GPR133/ADGRD1 agonist with an EC50 of 1.6 nM (293T cells). GPR133 agonist 1 activates GPR133, thereby regulating the downstream cAMP signaling pathway. GPR133 agonist 1 enhances muscle strength and endurance in mice. GPR133 agonist 1 can be used in research related to muscular atrophy, myasthenia, sarcopenia, erectile dysfunction, vestibular dysfunction, obesity, and non-alcoholic fatty liver disease[1].
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GPR133 agonist 1 | 99.87% | GPR133 agonist 1 is an orally active GPR133/ADGRD1 agonist with an EC50 of 1.6 nM (293T cells). GPR133 agonist 1 activates GPR133, thereby regulating the downstream cAMP signaling pathway. GPR133 agonist 1 enhances muscle strength and endurance in mice. GPR133 agonist 1 can be used in research related to muscular atrophy, myasthenia, sarcopenia, erectile dysfunction, vestibular dysfunction, obesity, and non-alcoholic fatty liver disease. | ||||||||||||||||||||
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