362512-81-0
362512-81-0
Chemical Structure
σ1 Receptor antagonist 4
- CAS No.: 362512-81-0
- Formula:C19H20FNO
- Molecular Weight:297.37
IUPAC Name: (3R,4R,7R,8R)-2-(3-fluorophenethyl)octahydro-1,3,4,6-(epiethane[1,1,2,2]tetrayl)pentaleno[1,6-bc]pyrrol-2a(2H)-ol
InChIKey: FYGREZKTJIXWIH-VLDSNRLISA-N
SMILES: OC12[C@H]3[C@@H]4C(C5C2C6[C@@H]3[C@H]4C5C6)N1CCC7=CC(F)=CC=C7
Biological Activity: σ1 Receptor antagonist 4 (compound TC1) is a selective sigma1 (σ1) receptor antagonist with a Ki of 10 nM. σ1 Receptor antagonist 4 is weakly active at σ2 receptor (Ki of 370 nM) and has no activity at dopamine (DAT), serotonin (SERT), and norepinephrine (NET) transporters[1].
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σ1 Receptor antagonist 4 | σ1 Receptor antagonist 4 (compound TC1) is a selective sigma1 (σ1) receptor antagonist with a Ki of 10 nM. σ1 Receptor antagonist 4 is weakly active at σ2 receptor (Ki of 370 nM) and has no activity at dopamine (DAT), serotonin (SERT), and norepinephrine (NET) transporters. | |||||||||||||||||||||
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