491611-43-9
491611-43-9
Chemical Structure
MRS2298
- CAS No.: 491611-43-9
- Formula:C10H16ClN5O8P2
- Molecular Weight:431.66
IUPAC Name: 2-((2-chloro-6-(methylamino)-9H-purin-9-yl)methyl)propane-1,3-diyl bis(dihydrogen phosphate)
InChIKey: GMCUIIHBWNOHIM-UHFFFAOYSA-N
SMILES: O=P(OCC(COP(O)(O)=O)CN1C=NC2=C(N=C(N=C12)Cl)NC)(O)O
Biological Activity: MRS2298? is a potent acyclic P2Y1 receptor antagonist with a Ki of 29.6 nM. MRS2298 inhibits the ADP-induced aggregation of human platelets with an IC50 of 62.8 nM. MRS2298 inhibits Ca2+ rise in platelets with an IC50 of 810 nM[1].
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MRS2298 | MRS2298? is a potent acyclic P2Y1 receptor antagonist with a Ki of 29.6 nM. MRS2298 inhibits the ADP-induced aggregation of human platelets with an IC50 of 62.8 nM. MRS2298 inhibits Ca2+ rise in platelets with an IC50 of 810 nM. | |||||||||||||||||||||
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