50330-93-3
50330-93-3
Chemical Structure
N-Desmethyl Rilmazolam
- CAS No.: 50330-93-3
- Formula:C18H13Cl2N5O
- Molecular Weight:386.23
InChIKey: PVNXUCAAXXYFKB-UHFFFAOYSA-N
SMILES: O=C(C1=NN(C2=C(C(C3=C(Cl)C=CC=C3)=NC4)C=C(Cl)C=C2)C4=N1)NC
Biological Activity: N-Desmethyl Rilmazolam is a metabolite of Rilmazolam (HY-150334) and 450191-S (HY-U00228). N-Desmethyl Rilmazolam significantly enhances the activity of 7-ethoxycoumarin O-deethylase. N-Desmethyl Rilmazolam can be used in insomnia-related studies[1][2].
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N-Desmethyl Rilmazolam | N-Desmethyl Rilmazolam is a metabolite of Rilmazolam (HY-150334) and 450191-S (HY-U00228). N-Desmethyl Rilmazolam significantly enhances the activity of 7-ethoxycoumarin O-deethylase. N-Desmethyl Rilmazolam can be used in insomnia-related studies. | |||||||||||||||||||||
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References
- [1]. Matsubara T, et al. Induction of rat liver microsomal drug-metabolizing enzymes by a new sleep inducer 450191-S and plasma levels of 450191-S-metabolites. Journal of pharmacobio-dynamics. 1986 Mar;9(3):249-56. [Content Brief]
- [2]. Kronstrand R, et al. Rilmazafone: A designer benzodiazepine pro-drug involved in fatal intoxications. Journal of analytical toxicology. 2023 Sep 15;47(7):640-643. [Content Brief]
