546141-08-6
546141-08-6
Chemical Structure
URB-597
Synonym(s): KDS-4103
- CAS No.: 546141-08-6
- Formula:C20H22N2O3
- Molecular Weight:338.40
IUPAC Name: 3'-carbamoyl-[1,1'-biphenyl]-3-yl cyclohexylcarbamate
InChIKey: ROFVXGGUISEHAM-UHFFFAOYSA-N
SMILES: O=C(OC1=CC(C2=CC=CC(C(N)=O)=C2)=CC=C1)NC3CCCCC3
Biological Activity: URB-597 (KDS-4103) is an orally bioavailable and selective FAAH inhibitor. URB-597 inhibits FAAH activity with an IC50s of approximately 5 nM in rat brain membranes, 0.5 nM in intact rat neurons, 3 nM in human liver microsomes. Antidepressant-like effects. Analgesic activity[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
URB-597 | 98.53% | URB-597 (KDS-4103) is an orally bioavailable and selective FAAH inhibitor. URB-597 inhibits FAAH activity with an IC50s of approximately 5 nM in rat brain membranes, 0.5 nM in intact rat neurons, 3 nM in human liver microsomes. Antidepressant-like effects. Analgesic activity. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
URB-597 (Standard) | ≥98% | URB-597 (Standard) is the analytical standard of URB-597. This product is intended for research and analytical applications. URB-597 (KDS-4103) is an orally bioavailable and selective FAAH inhibitor. URB-597 inhibits FAAH activity with an IC50s of approximately 5 nM in rat brain membranes, 0.5 nM in intact rat neurons, 3 nM in human liver microsomes. Antidepressant-like effects. Analgesic activity. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
