872002-73-8
Chemical Structure
WAY-207024 dihydrochloride
- CAS No.: 872002-73-8
- Formula:C30H34Cl2N6
- Molecular Weight:549.54
IUPAC Name: 6-((4-(2-(4-(tert-butyl)phenyl)-1H-benzo[d]imidazol-7-yl)piperazin-1-yl)methyl)quinoxaline dihydrochloride
InChIKey: REQCNTGYEABOIT-UHFFFAOYSA-N
SMILES: CC(C1=CC=C(C2=NC3=CC=CC(N4CCN(CC5=CC=C6N=CC=NC6=C5)CC4)=C3N2)C=C1)(C)C.[H]Cl.[H]Cl
Biological Activity: WAY-207024 dihydrochloride is an orally active gonadotropin releasing hormone receptor (GnRH-R) antagonist (human GnRH: IC50 of 12 nM, rat GnRH: IC50 of 71 nM). WAY-207024 dihydrochloride inhibits rat LH release with an IC50 of 350 nM. WAY-207024 dihydrochloride lowers rat plasma leuteinizing hormone (LH) levels after oral administration[1].
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WAY-207024 dihydrochloride | WAY-207024 dihydrochloride is an orally active gonadotropin releasing hormone receptor (GnRH-R) antagonist (human GnRH: IC50 of 12 nM, rat GnRH: IC50 of 71 nM). WAY-207024 dihydrochloride inhibits rat LH release with an IC50 of 350 nM. WAY-207024 dihydrochloride lowers rat plasma leuteinizing hormone (LH) levels after oral administration. | |||||||||||||||||||||
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