874882-72-1
874882-72-1
Chemical Structure
S(-)-Cyanopindolol hemifumarate
- CAS No.: 874882-72-1
- Formula:C16H21N3O2·1/2C4H4O4
- Molecular Weight:345.20
IUPAC Name: (S)-4-(3-(tert-butylamino)-2-hydroxypropoxy)-1H-indole-2-carbonitrile fumarate
SMILES: OC(/C=C/C(O)=O)=O.CC(C)(C)NC[C@H](O)COC1=C2C(NC(C#N)=C2)=CC=C1.[1/2]
Biological Activity: S(−)-Cyanopindolol hemifumarate is an isomer of Cyanopindolol (HY-W795507). S(-)-Cyanopindolol hemifumarate is a 5-HT1A/1B serotonin receptor antagonist and a β3-adrenoceptor antagonist[1][2].
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S(-)-Cyanopindolol hemifumarate | S(−)-Cyanopindolol hemifumarate is an isomer of Cyanopindolol (HY-W795507). S(-)-Cyanopindolol hemifumarate is a 5-HT1A/1B serotonin receptor antagonist and a β3-adrenoceptor antagonist. | |||||||||||||||||||||
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References
- [1]. Giles H, et al. Characterization of a 5-HT1B receptor on CHO cells: functional responses in the absence of radioligand binding. Br J Pharmacol. 1996 Mar;117(6):1119-26. [Content Brief]
- [2]. Hoey AJ, et al. Characteristics of cyanopindolol analogues active at the beta 3-adrenoceptor in rat ileum. Br J Pharmacol. 1996 Oct;119(3):564-8. [Content Brief]
