913344-84-0
913344-84-0
Chemical Structure
PF 02367982
- CAS No.: 913344-84-0
- Formula:C19H20N4O2
- Molecular Weight:336.39
IUPAC Name: 2-(4-(4-cyanophenoxy)-3,5-dicyclopropyl-1H-pyrazol-1-yl)-N-methylacetamide
InChIKey: PQGLAOODCQDRAR-UHFFFAOYSA-N
SMILES: O=C(NC)CN1N=C(C2CC2)C(OC3=CC=C(C#N)C=C3)=C1C4CC4
Biological Activity: PF 02367982 is a potent and select progesterone receptor (PR) antagonist with an IC50 value of 47.3 nM. PF 02367982 has oral activity[1].
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PF 02367982 | PF 02367982 is a potent and select progesterone receptor (PR) antagonist with an IC50 value of 47.3 nM. PF 02367982 has oral activity. | |||||||||||||||||||||
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References
- [1]. Alexander de Giorgio-Miller, et al. The translational pharmacology of a novel, potent, and selective nonsteroidal progesterone receptor antagonist, 2-[4-(4-cyano-phenoxy)-3,5-dicyclopropyl-1H-pyrazol-1-yl]-N-methylacetamide (PF-02367982). J Pharmacol Exp Ther. 2008 Oct;327(1):78-87. [Content Brief]
