934526-89-3
934526-89-3
Chemical Structure
Pilaralisib
Synonym(s): XL-147; SAR245408
- CAS No.: 934526-89-3
- Formula:C25H25ClN6O4S
- Molecular Weight:541.02
IUPAC Name: 2-amino-N-(3-(N-(3-((2-chloro-5-methoxyphenyl)amino)quinoxalin-2-yl)sulfamoyl)phenyl)-2-methylpropanamide
InChIKey: QINPEPAQOBZPOF-UHFFFAOYSA-N
SMILES: CC(C)(N)C(NC1=CC=CC(S(=O)(NC2=NC3=CC=CC=C3N=C2NC4=CC(OC)=CC=C4Cl)=O)=C1)=O
Biological Activity: Pilaralisib (XL147; SAR245408) is a potent and highly selective class I PI3Ks inhibitor with IC50s of 39 nM, 383 nM, 23 nM and 36 nM for PI3Kα, PI3Kβ, PI3Kγ, and PI3Kδ.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Pilaralisib | 98.81% | Pilaralisib (XL147; SAR245408) is a potent and highly selective class I PI3Ks inhibitor with IC50s of 39 nM, 383 nM, 23 nM and 36 nM for PI3Kα, PI3Kβ, PI3Kγ, and PI3Kδ. | ||||||||||||||||||||
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Pilaralisib (Standard) | ≥98% | Pilaralisib (Standard) is the analytical standard of Pilaralisib. This product is intended for research and analytical applications. Pilaralisib (XL147; SAR245408) is a potent and highly selective class I PI3Ks inhibitor with IC50s of 39 nM, 383 nM, 23 nM and 36 nM for PI3Kα, PI3Kβ, PI3Kγ, and PI3Kδ. | ||||||||||||||||||||
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