943344-76-1
Chemical Structure
SR-16157
Synonym(s): NSC 732011; HLX-801
- CAS No.: 943344-76-1
- Formula:C27H44N2O4S
- Molecular Weight:492.71
IUPAC Name: (7R,8S,9S,13R,14S,17R)-17-(2-(2-(diethylamino)ethoxy)ethyl)-7,13-dimethyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthren-3-yl sulfamate
InChIKey: ASNNHMZDKNSENI-FYUXVVBBSA-N
SMILES: O=S(OC1=CC=C2[C@@]3([H])CC[C@]4(C)[C@@H](CCOCCN(CC)CC)CC[C@@]4([H])[C@]3([H])[C@H](C)CC2=C1)(N)=O
Biological Activity: SR-16157 (NSC 732011; HLX-801) is a dual-action steroid sulfatase (STS) inhibitor (IC50 = 0.1 uM) and selective ERα modulator. SR-16157 exhibits STS inhibitory and anti-estrogenic effects in breast cancer cells. SR-16157 may be used in breast cancer research[1].
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SR-16157 | SR-16157 (NSC 732011; HLX-801) is a dual-action steroid sulfatase (STS) inhibitor (IC50 = 0.1 uM) and selective ERα modulator. SR-16157 exhibits STS inhibitory and anti-estrogenic effects in breast cancer cells. SR-16157 may be used in breast cancer research. | |||||||||||||||||||||
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