957054-30-7
957054-30-7
Chemical Structure
Pictilisib
Synonym(s): GDC-0941
- CAS No.: 957054-30-7
- Formula:C23H27N7O3S2
- Molecular Weight:513.64
IUPAC Name: 4-(2-(1H-indazol-4-yl)-6-((4-(methylsulfonyl)piperazin-1-yl)methyl)thieno[3,2-d]pyrimidin-4-yl)morpholine
InChIKey: LHNIIDJUOCFXAP-UHFFFAOYSA-N
SMILES: CS(N1CCN(CC2=CC3=C(C(N4CCOCC4)=NC(C5=CC=CC6=C5C=NN6)=N3)S2)CC1)(=O)=O
Biological Activity: Pictilisib (GDC-0941) is a potent inhibitor of PI3Kα/δ with an IC50 of 3 nM, with modest selectivity against p110β (11-fold) and p110γ (25-fold).
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
Pictilisib | 99.77% | Pictilisib (GDC-0941) is a potent inhibitor of PI3Kα/δ with an IC50 of 3 nM, with modest selectivity against p110β (11-fold) and p110γ (25-fold). | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
Pictilisib (Standard) | 98.06% | Pictilisib (Standard) is the analytical standard of Pictilisib. This product is intended for research and analytical applications. Pictilisib (GDC-0941) is a potent inhibitor of PI3Kα/δ with an IC50 of 3 nM, with modest selectivity against p110β (11-fold) and p110γ (25-fold). | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
