ERα ligand 2
ERα ligand 2 is a ligand for the PROTAC target protein ERα, which can be used to synthesis of ERα degraders (PROTACs), such as Vepdegestrant (HY-138642).
For research use only. We do not sell to patients.
- Formula: C22H20O
- Molecular Weight:300.39
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
[1]|
ERα |
In Vitro
PROTACs contain two different ligands connected by a linker; one is a ligand for an E3 ubiquitin ligase and the other is for the target protein. PROTACs exploit the intracellular ubiquitin-proteasome system to selectively degrade target proteins.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Molecular Weight 300.39
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Formula C22H20O
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SMILES
OC1=CC2=C([C@@H](C3=CC=CC=C3)[C@@H](C4=CC=CC=C4)CC2)C=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
ERα ligand 2 Related Classifications
HY-178077 Related Classifications
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