G2iA
G2iA is a selective GLUT2 inhibitor that inhibits GLUT2-mediated glucose transport with an IC50 of 0.61 µM.
For research use only. We do not sell to patients.
- CAS No.: 536702-12-2
- Formula: C27H24FN3O2S
- Molecular Weight:473.56
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Description
IC50 & Target
[1]|
GLUT2 0.61 μM (IC50) |
In Vitro
G2iA (100 µM; 10 min) is a GLUT2-selective inhibitor that, at a concentration of 100 µM, does not significantly inhibit GLUT1, GLUT3, GLUT4, or GLUT5 in hxt0 yeast transport assays[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 536702-12-2
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Molecular Weight 473.56
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Formula C27H24FN3O2S
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SMILES
O=C(CSC1=C(C)NC2=C1C=CC=C2)N3N=C(CC3C4=CC=C(C=C4)F)C5=CC=C(OC)C=C5
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)