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Cat. No.: HY-187976

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Melatonin receptor ligand-1

Melatonin receptor ligand-1 (compound AI-35) is a melatonin receptor ligand. Melatonin receptor ligand-1 has an IC₅₀ of 1020 nM and a K_i of 289 nM at the quail target.

For research use only. We do not sell to patients.

CAS No.: 214416-49-6
Formula: C₁₄H₁₈N₂O₃
Molecular Weight:262.30

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Melatonin receptor ligand-1 Chemical Structure

CAS No.: 214416-49-6

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- In Vitro
Chemical Information
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Biological Activity

Description

Melatonin receptor ligand-1 (compound AI-35) is a melatonin receptor ligand. Melatonin receptor ligand-1 has an IC₅₀ of 1020 nM and a K_i of 289 nM at the quail target^[1].

All Melatonin Receptor Isoforms :

In Vitro

Melatonin receptor ligand-1 (compound AI-35) displaces 2-[¹²⁵I]-iodomelatonin with an IC₅₀ of 1020 nM and a K_i of 289 nM in quail optic tectum membrane binding assays^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 214416-49-6
Molecular Weight 262.30
Formula C₁₄H₁₈N₂O₃
SMILES

O=C(C)NCCC1=CNC2=C1C=C(OCCO)C=C2
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Mor M, et al. Melatonin receptor ligands: synthesis of new melatonin derivatives and comprehensive comparative molecular field analysis (CoMFA) study. Journal of medicinal chemistry. 1998 Sep 24;41(20):3831-44.

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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