Sulfonimidamides as sulfonamides bioisosteres: rational evaluation through synthetic, in vitro, and in vivo studies with γ-secretase inhibitors

  • ChemMedChem. 2012 Mar 5;7(3):396-9. doi: 10.1002/cmdc.201200014.
Fernando Sehgelmeble  1 ,  Juliette Janson ,  Colin Ray ,  Susanne Rosqvist ,  Susanne Gustavsson ,  Linda I Nilsson ,  Alexander Minidis ,  Jörg Holenz ,  Didier Rotticci ,  Johan Lundkvist ,  Per I Arvidsson
Affiliations
  • 1. Medicinal Chemistry, iScience, CNSP iMed, AstraZeneca R&D Södertälje, Västra Mälarehamnen 9, 15185 Södertälje, Sweden.
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