1 Result for "

A286501

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "A286501" in MCE Product Catalog:

Cat. No.: HY-116005
CAS No.: 483341-15-7
A-286501 is an orally active adenosine kinase inhibitor with an IC50 of 0.47 nM (rat brain cytosol). A-286501 blocks the phosphorylation of adenosine to AMP and increases adenosine. A-286501 mediates non-opioid adenosine receptor-dependent antinociceptive and anti-inflammatory effects, reduces paw edema, myeloperoxidase activity, and tactile allodynia, and produces antinociceptive effects in acute, inflammatory, neuropathic, and hyperalgesic models. A-286501 can be used in research on inflammatory pain, neuropathic pain, and diabetic neuropathy .
loading...
    loading...