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FK3657

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Cat. No.: HY-15791
CAS No.: 167838-64-4
Synonyms: FK-3657
FR173657 (FK-3657) is an orally active, selective bradykinin B2 receptor antagonist. FR173657 induces Apoptosis, G0/G1 phase arrest, and p38 MAPK/p27Kip1 signaling. FR173657 blocks afferent neuron activation, tumor vascular hyperpermeability, tumor angiogenesis/growth, colorectal proliferation, kinin-mediated invasion/migration, and airway plasma extravasation. FR173657 can be used in research on inflammatory pain, asthma, triple-negative breast cancer, psoriasis, pancreatitis, acute cystitis, skin inflammation, sarcoma 180, colorectal liver metastasis, and Carrageenan-induced pleurisy .
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