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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
1 Result for "
MK1421
" in MedChemExpress (MCE) Product Catalog:
Products (1)
1 Results for "MK1421" in MCE Product Catalog:
Cat. No.: HY-12819
CAS No.: 1235995-16-0
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MK-1421 is an orally active sstr3 antagonist. MK-1421 inhibits sstr3 with IC50 values of 2.3 nM (human), 1.3 nM (mouse), 0.6 nM (rat), 2.5 nM (dog), and 1.0 nM (rhesus monkey). MK-1421 inhibits hERG (human IC50 32.2 μM). MK-1421 dose-dependently reduces blood glucose fluctuations and enhances insulin secretion under high glucose conditions but not low glucose conditions, without affecting glucagon or somatostatin release. MK-1421 can be used for research on type 2 diabetes .
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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
