17

17 Publications Verification

CAS No.: 20449-79-0

Target:

Research Areas:

Melittin is a PLA₂ activator, stimulates the activity of the low molecular weight PLA₂, while it does not the increase activity of the high molecular weight PLA₂ .

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17

Melittin TFA

17 Publications Verification

Cat. No.: HY-P0233A

Target:

Phospholipase

Research Areas:

Infection Cancer

Melittin TFA is a PLA₂ activator, stimulates the activity of the low molecular weight PLA₂, while it does not the increase activity of the high molecular weight PLA₂ .

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8

Darapladib

8 Cited Publications

Cat. No.: HY-10521

CAS No.: 356057-34-6

Purity: 99.94%

Synonyms: SB-480848

Target:

Phospholipase Apoptosis

Research Areas:

Cardiovascular Disease Cancer

Darapladib (SB-480848) is an orally active, selective and reversible Lp-PLA2 inhibitor (IC₅₀=0.25 nM). Darapladib can trigger irreversible actions on glioma cell apoptosis and induce cycle arrest. Darapladib can be used in the study of atherosclerosis and cancer .

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8

(E/Z)-BML264

8 Cited Publications

Cat. No.: HY-118628

CAS No.: 110683-10-8

Purity: 99.63%

Synonyms: N-(p-Amylcinnamoyl) anthranilic acid; ACA

Target:

Phospholipase TRP Channel

Research Areas:

Cardiovascular Disease

(E/Z)-BML264 (N-(p-amylcinnamoyl) Anthranilic Acid) is a broad spectrum Phospholipase A₂ (PLA₂) inhibitor and TRP channel blocker . (E/Z)-BML264 is a SLC13A3 inhibitor. (E/Z)-BML264 (N-(p-amylcinnamoyl) Anthranilic Acid) is also an effective reversible inhibitor of calcium-activated chloride channels, has potential to treat arrhythmia .

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7

Azoramide

7 Cited Publications

Cat. No.: HY-18705

CAS No.: 932986-18-0

Target:

Apoptosis Reactive Oxygen Species (ROS) Caspase Bcl-2 Family Mitochondrial Metabolism

Research Areas:

Endocrinology

Azoramide is a potent, orally active small-molecule modulator of the unfolded protein response (UPR). Azoramide improves ER protein folding and elevates ER chaperone capacity, which together protects cells against ER stress. Azoramide alleviates PLA2G6 mutant-induced ER stress through modulating unfolded protein response, and enhances the CERB signaling to rescue mitochondrial function, thereby preventing apoptosis of DA neurons. Azoramide has antidiabetic activity .

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3

PLA2G2A Protein, Mouse (P.pastoris, His)

3 Cited Publications

Cat. No.: HY-P74628

Purity: ≥ 95%, as determined by reducing SDS-PAGE.

Synonyms: PLA2G2A; Non-Pancreatic Secretory Phospholipase A2; Prev. PLA2B; Phospholipase A2; Prev. PLA2L; RASF-A; Phosphatidylcholine 2-Acylhydrolase 2A; PLA2S; Phospholipase A2, Membrane Associated; PLAS1; Group IIA Phospholipase A2; SPLA2; GIIC SPLA2; MOM1; Phosp

Species:

Mouse

Source:

P. pastoris

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3

Rilapladib

3 Cited Publications

Cat. No.: HY-102004

CAS No.: 412950-08-4

Purity: 99.44%

Synonyms: SB 659032

Target:

Phospholipase

Research Areas:

Neurological Disease Inflammation/Immunology

Rilapladib (SB 659032) is a selective Lp-PLA₂ (lipoprotein-associated phospholipase A₂) inhibitor with an IC₅₀ of 230 pM . Rilapladib (SB 659032) is also a PAFR (Platelet Activating Factor Receptor) antagonist .

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2

1-Naphthaleneacetic acid

2 Cited Publications

Cat. No.: HY-18570

CAS No.: 86-87-3

Synonyms: 1-Naphthylacetic acid

1-Naphthaleneacetic acid (1-Naphthylacetic acid), a auxin, can promote plant growth. 1-Naphthaleneacetic acid is also an inhibitor of PLA₂, with an IC₅₀ of 13.16 μM .

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2

1-Naphthaleneacetic acid potassium salt

2 Cited Publications

Cat. No.: HY-18570A

CAS No.: 15165-79-4

Synonyms: Potassium 1-Naphthaleneacetate

Target:

Environmental Pollutants Phospholipase

Research Areas:

Others

1-Naphthaleneacetic acid potassium salt (Potassium 1-Naphthaleneacetate), a synthetic auxin, can promote plant growth. 1-Naphthaleneacetic acid potassium salt is also an inhibitor of PLA₂, with an IC₅₀ of 13.16 μM .

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