1 Result for "

Rockout

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "Rockout" in MCE Product Catalog:

Cat. No.: HY-112362
CAS No.: 7272-84-6
Purity:  ≥99.0%
Synonyms: Rockout; 3-(4-Pyridinyl)-1H-indole; Rho Kinase Inhibitor III, Rockout
Target:  

ROCK Actin

Research Areas:  

Inflammation/Immunology

3-(4-Pyridyl)indole (Rockout; 3-(4-Pyridinyl)-1H-indole; Rho Kinase Inhibitor III, Rockout) is a Rho-kinase inhibitor (IC50 = 25 μM). 3-(4-Pyridyl)indole inhibits cell migration, membrane blebbing, and stress fiber and focal adhesion formation, and induces actin stress fiber disassembly. 3-(4-Pyridyl)indole promotes cell spreading and alters cell morphology and dynamics. 3-(4-Pyridyl)indole inhibits PRK2. 3-(4-Pyridyl)indole is used in wound healing research .
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