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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
12 Results for "
SSTR3
" in MedChemExpress (MCE) Product Catalog:
Products (12)
12 Results for "SSTR3" in MCE Product Catalog:
6
6 Cited Publications
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MK-4256 is a potent and selective SSTR3 antagonist with IC50s of 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively.
Cat. No.: HY-177493
CAS No.: 3086695-73-7
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SSTR3 Agonist-1 (Compound EX 38) is an orally active SSTR3 agonist, with an EC50 of 0.14 nM. SSTR3 Agonist-1 reduces the kidney cystic index. SSTR3 Agonist-1 can be used in the research of autosomal dominant polycystic kidney disease .
Cat. No.: HY-177493A
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SSTR3 agonist-1 TFA is a potent, orally active, and selective SSTR3 agnoist (EC50 =0.14 nM). SSTR3 agonist-1 TFA binds to SSTR3 receptor to inhibit cAMP activity. SSTR3 agonist-1 TFA decreases kidney weight and kidney cystic index (KCI) in a mouse model of autosomal dominant polycystic kidney disease (ADPKD). SSTR3 agonist-1 TFA can be used for ADPKD research .
Cat. No.: HY-RS13826
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SSTR3 Human Pre-designed siRNA Set A contains three designed siRNAs for SSTR3 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS13827
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Sstr3 Mouse Pre-designed siRNA Set A contains three designed siRNAs for Sstr3 gene (Mouse), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS13828
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Sstr3 Rat Pre-designed siRNA Set A contains three designed siRNAs for Sstr3 gene (Rat), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-P3618
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Cat. No.: HY-12819
CAS No.: 1235995-16-0
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MK-1421 is an orally active sstr3 antagonist. MK-1421 inhibits sstr3 with IC50 values of 2.3 nM (human), 1.3 nM (mouse), 0.6 nM (rat), 2.5 nM (dog), and 1.0 nM (rhesus monkey). MK-1421 inhibits hERG (human IC50 32.2 μM). MK-1421 dose-dependently reduces blood glucose fluctuations and enhances insulin secretion under high glucose conditions but not low glucose conditions, without affecting glucagon or somatostatin release. MK-1421 can be used for research on type 2 diabetes .
Cat. No.: HY-P4555
CAS No.: 340821-13-8
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Cat. No.: HY-P2434
CAS No.: 846569-60-6
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Cat. No.: HY-P2150
CAS No.: 1815618-17-7
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
