42 Results for "

cholinergic agent

" in MedChemExpress (MCE) Product Catalog:
Products (42)

42 Results for "cholinergic agent" in MCE Product Catalog:

4
Pyrantel pamoate
Pyrantel pamoate
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4 Cited Publications
Cat. No.: HY-12640
CAS No.: 22204-24-6
Purity:  99.97%
Synonyms: Pyrantel embonate
Target:  

Parasite nAChR

Research Areas:  

Infection

Pyrantel pamoate is an orally active antiparasitic agent. Pyrantel pamoate induces spastic paralysis in parasites via actions on neural and muscular cholinergic receptors as a nicotinic acetylcholine receptor (nAChR) agonist. Pyrantel pamoate eliminates both immature and mature endoparasites in horses. Pyrantel pamoate can be used in research related to parasitic infections .
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Rivastigmine
Rivastigmine
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1 Cited Publications
Cat. No.: HY-17368
CAS No.: 123441-03-2
Synonyms: ENA 713 free base; SDZ-ENA 713 free base
Target:  

Cholinesterase (ChE)

Research Areas:  

Neurological Disease

Rivastigmine (ENA 713 free base) is an orally active and potent cholinesterase (ChE) inhibitor and inhibits butyrylcholinesterase (BChE) and acetylcholinesteras (AChE) with IC50s of 0.037 μM , 4.15 μM, respectively. Rivastigmine can pass the blood brain barrier (BBB). Rivastigmine is a parasympathomimetic or cholinergic agent used for the research of mild to moderate dementia of the Alzheimer's type and dementia due to Parkinson's disease .
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Rivastigmine tartrate
Rivastigmine tartrate
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1 Cited Publications
Cat. No.: HY-11017
CAS No.: 129101-54-8
Purity:  99.03%
Synonyms: ENA 713; SDZ-ENA 713
Target:  

Cholinesterase (ChE)

Research Areas:  

Neurological Disease

Rivastigmine tartrate (ENA 713; SDZ-ENA 713) is an orally active and potent cholinesterase (ChE) inhibitor and inhibits butyrylcholinesterase (BChE) and acetylcholinesteras (AChE) with IC50s of 0.037 μM, 4.15 μM, respectively. Rivastigmine tartrate can pass the blood brain barrier (BBB). Rivastigmine tartrate is a parasympathomimetic or cholinergic agent used for the research of mild to moderate dementia of the Alzheimer's type and dementia due to Parkinson's disease .
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Pyrantel tartrate
Pyrantel tartrate
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1 Cited Publications
Cat. No.: HY-12641
CAS No.: 33401-94-4
Purity:  98.69%
Target:  

Parasite nAChR

Research Areas:  

Infection

Pyrantel tartrate is an orally active antiparasitic agent. Pyrantel tartrate induces spastic paralysis in parasites via actions on neural and muscular cholinergic receptors as a nicotinic acetylcholine receptor (nAChR) agonist. Pyrantel tartrate eliminates both immature and mature endoparasites in horses. Pyrantel tartrate can be used in research related to parasitic infections .
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Dicyclomine hydrochloride
Dicyclomine hydrochloride
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Cat. No.: HY-B1339
CAS No.: 67-92-5
Synonyms: Dicycloverine hydrochloride
Target:  

mAChR

Research Areas:  

Neurological Disease

Dicyclomine hydrochloride is a potent and orally active muscarinic cholinergic receptors antagonist. Dicyclomine hydrochloride shows high affinity for muscarinic M1 receptor subtype (Ki=5.1 nM) and M2 receptor subtype (Ki=54.6 nM) in brush-border membrane and basal plasma membranes, respectively . Dicyclomine is an antispasmodic agent and relieves smooth muscle spasm of the gastrointestinal tract in vivo .
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Pyrantel pamoate (Standard)
Pyrantel pamoate (Standard)
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Cat. No.: HY-12640R
CAS No.: 22204-24-6
Synonyms: Pyrantel embonate (Standard)
Target:  

Reference Standards Parasite nAChR

Research Areas:  

Infection

Pyrantel pamoate (Standard) (Pyrantel embonate (Standard)) is the analytical standard of Pyrantel pamoate (HY-12640). This product is intended for research and analytical applications. Pyrantel pamoate is an orally active antiparasitic agent. Pyrantel pamoate induces spastic paralysis in parasites via actions on neural and muscular cholinergic receptors as a nicotinic acetylcholine receptor (nAChR) agonist. Pyrantel pamoate eliminates both immature and mature endoparasites in horses. Pyrantel pamoate can be used in research related to parasitic infections .
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Carpronium chloride
Carpronium chloride
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Cat. No.: HY-B2198
CAS No.: 13254-33-6
Synonyms: Actinomin chloride
Target:  

Cholinesterase (ChE)

Research Areas:  

Neurological Disease

Carpronium (Actinomin) chloride is an orally active cholinergic agonist, local vasodilator and parasympathomimetic agent. Carpronium chloride is structurally similar to acetylcholine. Carpronium chloride promotes hair growth, and oral overdose induces cholinergic crisis. Carpronium chloride is applicable to research related to alopecia areata .
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Z-4105
Z-4105
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Cat. No.: HY-W987949
CAS No.: 119737-52-9
Target:  

Others

Research Areas:  

Neurological Disease

Z-4105 is an orally active nootropic agent. Z-4105 reverses the amnesic effects of electroconvulsive shock (ECS) and methylazoxymethanol acetate (MAM), and improves learning and memory functions. Z-4105 enhances the activity of the brain cholinergic system without affecting other neurotransmitter systems. Z-4105 significantly alleviates neuropathic pain in rats. Z-4105 can be used in the research of neuropathic pain and brain dysfunction .
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Rivastigmine (Standard)
Rivastigmine (Standard)
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Cat. No.: HY-17368R
CAS No.: 123441-03-2
Synonyms: ENA 713 free base(Standard); SDZ-ENA 713 free base(Standard)
Target:  

Reference Standards Cholinesterase (ChE)

Research Areas:  

Neurological Disease

Rivastigmine (Standard) is the analytical standard of Rivastigmine. This product is intended for research and analytical applications. Rivastigmine (ENA 713 free base) is an orally active and potent cholinesterase (ChE) inhibitor and inhibits butyrylcholinesterase (BChE) and acetylcholinesteras (AChE) with IC50s of 0.037 μM , 4.15 μM, respectively. Rivastigmine can pass the blood brain barrier (BBB). Rivastigmine is a parasympathomimetic or cholinergic agent used for the research of mild to moderate dementia of the Alzheimer's type and dementia due to Parkinson's disease .
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Eucatropine
Eucatropine
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Cat. No.: HY-117284
CAS No.: 100-91-4
Target:  

mAChR

Research Areas:  

Neurological Disease

Eucatropine is a potent muscarinic acetylcholine receptor (mAChR) inhibitor with an IC50 value of 0.583 μM. Eucatropine acts as an anticholinergic agent. Eucatropine produces behavioral effects via central cholinergic receptive sites in cats .
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Caramiphen (edisylate)
Caramiphen (edisylate)
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Cat. No.: HY-B1585B
CAS No.: 125-86-0
Synonyms: Parpanil (edisylate)
Target:  

iGluR

Research Areas:  

Neurological Disease

Caramiphen edisylate (Parpanil edisylate) is an anticholinergic agent with NMDA receptor antagonist activity. Caramiphen edisylate can be used to inhibit diseases related to cholinergic neurotransmission. Caramiphen edisylate exerts its pharmacological effects by blocking cholinergic effects .
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Pyrantel
Pyrantel
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Cat. No.: HY-12641A
CAS No.: 15686-83-6
Target:  

Parasite nAChR

Research Areas:  

Infection

Pyrantel is an orally active antiparasitic agent. Pyrantel induces spastic paralysis in parasites via actions on neural and muscular cholinergic receptors as a nicotinic acetylcholine receptor (nAChR) agonist. Pyrantel eliminates both immature and mature endoparasites in horses. Pyrantel can be used in research related to parasitic infections .
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Dicyclomine
Dicyclomine
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Cat. No.: HY-B1339A
CAS No.: 77-19-0
Synonyms: Dicycloverine
Target:  

mAChR

Research Areas:  

Neurological Disease

Dicyclomine (Dicycloverine) is a potent and orally active muscarinic cholinergic receptors antagonist. Dicyclomine (Dicycloverine) shows high affinity for muscarinic M1 receptor subtype (Ki=5.1 nM) and M2 receptor subtype (Ki=54.6 nM) in brush-border membrane and basal plasma membranes, respectively . Dicyclomine is an antispasmodic agent and relieves smooth muscle spasm of the gastrointestinal tract in vivo .
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Trimedoxime
Trimedoxime
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Cat. No.: HY-165600A
CAS No.: 56-97-3
Synonyms: TMB-4
Target:  

Cholinesterase (ChE)

Research Areas:  

Others

Trimedoxime (TMB-4) is a blood-brain barrier-permeable cholinesterase reactivator . Trimedoxime reactivates cholinesterase inhibited by paraoxon, sarin, tabun and other agents, restricts the breakdown of acetylcholine and alleviates excessive cholinergic stimulation. Trimedoxime reduces mortality and prolongs survival time. Trimedoxime exhibits reactivation efficacy against AChE in rat tissues. Trimedoxime can be used in research related to organophosphate (paraoxon) poisoning and tabun poisoning .
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Pozanicline
Pozanicline
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Cat. No.: HY-14565
CAS No.: 161417-03-4
Synonyms: ABT-089
Target:  

nAChR

Research Areas:  

Neurological Disease

Pozanicline (ABT-089) selectively activate neuronal nicotinic acetylcholine receptor (nAChR) subtypes, is a novel cholinergic agent that is a partial agonist at α4β2* nAChRs (Ki=16 nM) and shows high selectivity for α6β2* and α4α5β2 nAChR subtypes, the binding affinity (Ki, rat) for Pozanicline to [ 3H] cytisine sites is 16.7 nM. Pozanicline reverses nicotine withdrawal-induced cognitive deficits, may be an effective component of novel therapeutic strategies for nicotine addiction .
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Caramiphen
Caramiphen
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Cat. No.: HY-B1585
CAS No.: 77-22-5
Synonyms: Parpanil
Target:  

iGluR

Research Areas:  

Neurological Disease

Parpanil is an anticholinergic agent with NMDA receptor antagonist activity. Parpanil can be used to inhibit diseases related to cholinergic neurotransmission. Parpanil exerts its pharmacological effects by blocking cholinergic effects .
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Ilmetropium iodide
Ilmetropium iodide
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Cat. No.: HY-109006
CAS No.: 129109-88-2
Target:  

mAChR

Research Areas:  

Neurological Disease

Ilmetropium iodide is an anticholinergic agent. Ilmetropium iodide selectively blocks M-cholinergic receptors of bronchial muscle, reduces or prevents bronchoconstrictor response associated with both cholinergic stimulation, as well as the impact of the factors that provoke bronchospasm. Strength and selectivity of ilmetropium iodide action substantially exceeds Atropine sulfate (HY-B1205A) and Ipratropium bromide (HY-B0241) .
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Doxacurium chloride
Doxacurium chloride
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Cat. No.: HY-A0215
CAS No.: 106819-53-8
Synonyms: BW-A 938U; Nuromax
Target:  

nAChR

Research Areas:  

Neurological Disease

Doxacurium chloride (BW A938U) is a potent non-depolarizing neuromuscular blocking agent. Doxacurium chloride binds to cholinergic receptors to antagonize acetylcholine, resulting in a block of neuromuscular transmission. Doxacurium chloride can be used for the research of neurological diseases .
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Suffruticosol A
Suffruticosol A
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Cat. No.: HY-N11872
CAS No.: 220936-82-3
Category:  

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