STK3-IN-1
STK3-IN-1 is an ATP-binding site inhibitor of STK3. STK3-IN-1 blocks the enzymatic activity of STK3 with an IC50 of 3.52 nM. STK3-IN-1 also exhibits inhibitory activity against STK4, a homolog closely related to STK3, with an IC50 of 14.73 nM.
For research use only. We do not sell to patients.
- Formula: C24H28N4O5
- Molecular Weight:452.50
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Description
IC50 & Target
[1]|
STK3 3.52 nM (IC50) |
STK3 14.73 nM (IC50) |
In Vitro
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
Molecular Weight 452.50
-
Formula C24H28N4O5
-
SMILES
OC1=CC(OCCOC(NC(C)(C)C)=O)=CC=C1C2=NC(N)=NC=C2C3=C(OC)C=CC=C3
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)