country

Change Language

EN - English
FR - Français
DE - Deutsch
ES - Español
JA - 日本語
KO - 한국어

Country or Region:

United States

Product Name	Size / Unit Price	Qty

Total: USD 0.00 Checkout

Cat. No.: HY-133722

Copy Link Print Information

ZAPA

ZAPA is a competitive GABA_C receptor antagonist.

For research use only. We do not sell to patients.

CAS No.: 92138-10-8
Formula: C₄H₆N₂O₂S
Molecular Weight:146.16

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

ZAPA Chemical Structure

CAS No.: 92138-10-8

Price

Stock

Quantity

Amount: USD 0.00

* Please select Quantity before adding items.

Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
- In Vitro
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

Description

ZAPA is a competitive GABA_C receptor antagonist^[1].

IC₅₀ & Target

^[1]

GABAC

In Vitro

ZAPA (compound 63) is a moderately potent competitive GABA_C receptor antagonist acting on poly (A)⁺ RNA from bovine retina expressed in Xenopus oocytes, with a K_B of 19 µM^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 92138-10-8
Molecular Weight 146.16
Formula C₄H₆N₂O₂S
SMILES

C(=C\C(O)=O)\SC(=N)N
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Chebib M, et al. GABA-Activated ligand gated ion channels: medicinal chemistry and molecular biology. J Med Chem. 2000 Apr 20;43(8):1427-47. [Content Brief]

Calculators

Molarity Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Dilution Calculator

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

Keywords

MOQ

Minimum order quantity

100 mg

Get Quote In-stock

Other size

Get Quote