1380585-51-2
1380585-51-2
Chemical Structure
CCBT-T-226
- CAS No.: 1380585-51-2
- Formula:C15H19N3O4S
- Molecular Weight:337.39
InChIKey: BBEFFOPCSBTRBM-UHFFFAOYSA-N
SMILES: O=C(C1=C(CCC)SC(NC(CC2=C(C)ON=C2C)=O)=N1)OC
Biological Activity: CCBT-T-226 is a BRD4-BD2 inhibitor with a Kd of 1.3 μM. CCBT-T-226 binds the conserved acetyl-lysine recognition site of BRD4-BD1 with reduced affinity. CCBT-T-226 has a Kd of 9 μM for BRD4-BD1. CCBT-T-226 exhibits domain selectivity for BRD4-BD2 over BRD4-BD1[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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CCBT-T-226 | CCBT-T-226 is a BRD4-BD2 inhibitor with a Kd of 1.3 μM. CCBT-T-226 binds the conserved acetyl-lysine recognition site of BRD4-BD1 with reduced affinity. CCBT-T-226 has a Kd of 9 μM for BRD4-BD1. CCBT-T-226 exhibits domain selectivity for BRD4-BD2 over BRD4-BD1. | |||||||||||||||||||||
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