2495322-59-1
2495322-59-1
Chemical Structure
CREBBP/EP300-IN-1
- CAS No.: 2495322-59-1
- Formula:C28H32ClN7O
- Molecular Weight:518.06
IUPAC Name: 6-chloro-N-((1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl)-N-methyl-2-(6-methyl-5-((1-methylazetidin-3-yl)amino)pyridin-2-yl)quinoline-4-carboxamide
InChIKey: GYCCIEWETQNUJP-UHFFFAOYSA-N
SMILES: O=C(C1=CC(=NC=2C=CC(Cl)=CC21)C=3N=C(C(=CC3)NC4CN(C)C4)C)N(C)CC=5C=NN(C5C)CC
Biological Activity: CREBBP/EP300-IN-1 is an inhibitor of CREBBP and EP300, with IC50 values of 0.01707 and 0.0065 μM, respectively. CREBBP/EP300-IN-1 exhibits anticancer activity against bladder cancer[1].
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CREBBP/EP300-IN-1 | CREBBP/EP300-IN-1 is an inhibitor of CREBBP and EP300, with IC50 values of 0.01707 and 0.0065 μM, respectively. CREBBP/EP300-IN-1 exhibits anticancer activity against bladder cancer. | |||||||||||||||||||||
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