CREBBP/EP300-IN-1
CREBBP/EP300-IN-1 is an inhibitor of CREBBP and EP300, with IC50 values of 0.01707 and 0.0065 μM, respectively. CREBBP/EP300-IN-1 exhibits anticancer activity against bladder cancer.
For research use only. We do not sell to patients.
- CAS No.: 2495322-59-1
- Formula: C28H32ClN7O
- Molecular Weight:518.06
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
[1]|
EP300 0.0065 μM (IC50) |
CREBBP 0.01707 μM (IC50) |
In Vitro
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2495322-59-1
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Molecular Weight 518.06
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Formula C28H32ClN7O
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SMILES
O=C(C1=CC(=NC=2C=CC(Cl)=CC21)C=3N=C(C(=CC3)NC4CN(C)C4)C)N(C)CC=5C=NN(C5C)CC
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CREBBP/EP300-IN-1 Related Classifications
HY-134516 Related Classifications
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