(Rac)-VU0637120
(Rac)-VU0637120 is the racemate of (S)-VU0637120 (HY-165125). (S)-VU0637120 is a selective Y4R antagonist that effectively reduces the binding of its endogenous ligand pancreatic polypeptide (PP) to Y4R, with an IC50 value of 2.7 μM. (S)-VU0637120 binds to an allosteric site of Y4R, which is located in the core region of the transmembrane structure of Y4R, near the binding pocket of pancreatic polypeptide (PP), with a KB of 380 nM. (Rac)-VU0637120 can be used for research on metabolic diseases.
For research use only. We do not sell to patients.
- CAS No.: 1214099-39-4
- Formula: C16H19N3O5S2
- Molecular Weight:397.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
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All Neuropeptide Y Receptor Isoforms
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Biological Activity
Description
Chemical Information
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CAS No. 1214099-39-4
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Molecular Weight 397.47
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Formula C16H19N3O5S2
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SMILES
O=C(C1N(S(=O)(C)=O)CCCC1)NC2=NC3=C(S2)C=C4OCCOC4=C3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
(Rac)-VU0637120 Related Classifications
HY-165125A Related Classifications
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