![[Des-Arg9]-Bradykinin acetate](https://file.medchemexpress.com/product_pic/hy-p0298a.gif "Click to View [Des-Arg9]-Bradykinin acetate Product Detail")
Scientific Reviews
Product Guides
Blogs
Topics
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
866 Results for "
B2
" in MedChemExpress (MCE) Product Catalog:
Products (866)
866 Results for "B2" in MCE Product Catalog:
20
Category:
Other Families Extract Plant Flavonoids Functional Molecules Research of Health Products Phenols Polyphenols Disease Research Fields Biflavones Cancer
Target:
17
17 Cited Publications
Synonyms: APTA-2217; BYK 20869; B9302-107
Target:
Research Areas:
Roflumilast (APTA-2217) is a selective PDE4 inhibitor with IC50s of 0.7, 0.9, 0.7, and 0.2 nM for PDE4A1, PDE4A4, PDE4B1, and PDE4B2, respectively, without affecting PDE1, PDE2, PDE3 or PDE5 isoenzymes from various cells.
14
Target:
Research Areas:
14
14 Cited Publications
Synonyms: HOE 140 acetate
Target:
Research Areas:
12
6
6 Cited Publications
Cat. No.: HY-N0604
CAS No.: 63223-86-9
Synonyms: Prosapogenin A2; Sanchinoside B2; Sanchinoside Rh1
6
Target:
Research Areas:
NSC 663284 (DA-3003-1) is a potent, cell-permeable, and irreversible Cdc25 dual specificity phosphatase inhibitor, has an IC50 for Cdc25B2 of 0.21 μM. NSC 663284 exhibits mixed competitive kinetics against Cdc25A, Cdc25B(2), and Cdc25C with Ki values of 29, 95, and 89 nM, respectively . NSC 663284 inhibits NSD2 (IC50 of 170 nM) through a direct interaction with the catalytic SET domain (Kd of 370 nM) [2].
4
4 Cited Publications
Cat. No.: HY-N0044
CAS No.: 52286-59-6
Synonyms: Ginsenoside B2; Panaxoside Re; Sanchinoside Re
Category:
Triterpenes Plant Neurological Disease Terpenoids Panax ginseng C. A. Meyer Extract Endogenous metabolite Disease Research Fields Cancer Araliaceae Extract
Target:
4
4 Cited Publications
Target:
Research Areas:
KM91104 is a cell-permeable V-ATPase a3-b2 inhibitor (IC50 = 2.3 µM). KM91104 reduces the metabolic activity, cell proliferation capacity and V-ATPase subunit protein expression levels of primary human hepatic stellate cells, increases intracellular ATP levels and decreases cytoplasmic pH. KM91104 reduces TLR4 expression on the surface of oligodendrocyte precursor cells, blocks the ENV-TLR4 interaction, and reverses oligodendrocyte myelination defects induced by ENV protein [2].
4
4 Cited Publications
4
Target:
Research Areas:
Osilodrostat (LCI699) is a potent, orally active11β-hydroxylase (CYP11B1) inhibitor with an IC50 value of 35 nM. Osilodrostat is a potent, orally aldosterone synthase (CYP11B2) inhibitor with IC50 values of 0.7 nM and 160 nM for human aldosterone synthase and rat aldosterone synthase, respectively. Osilodrostat inhibits aldosterone and corticosterone synthesis. Osilodrostat has blood pressure lowering ability. Osilodrostat can be used for research of Cushing syndrome (CS) [2] .
4
Target:
Research Areas:
Osilodrostat (LCI699) phosphate is a potent, orally active11β-hydroxylase (CYP11B1) inhibitor with an IC50 value of 35 nM. Osilodrostat phosphate is a potent, orally aldosterone synthase (CYP11B2) inhibitor with IC50 values of 0.7 nM and 160 nM for human aldosterone synthase and rat aldosterone synthase, respectively. Osilodrostat phosphate inhibits aldosterone and corticosterone synthesis. Osilodrostat phosphate has blood pressure lowering ability. Osilodrostat phosphate can be used for research of Cushing syndrome (CS) [2] .
3
3 Cited Publications
Synonyms: Riboflavine phosphate sodium; Riboflavin 5'-phosphate sodium; Riboflavine 5'-phosphate sodium
Target:
3
3 Cited Publications
Cat. No.: HY-N0652
CAS No.: 82373-94-2
Synonyms: 2,3,4',5-Tetrahydroxystilbene 2-O-D-glucoside
3
Target:
Research Areas:
Diethylstilbestrol is a non-steroidal female hormone that has oral activity and can act on menopausal and postmenopausal disorders. Diethylstilbestrol can induce DNA oxidation and Apoptosis of spermatogonial stem cells. Diethylstilbestrol can induce thymocyte Autophagy Diethylstilbestrol is a 11β-hydroxysteroid dehydrogenase 2 (HSD11B2) inhibitor. [2] .
2
2 Cited Publications
Cat. No.: HY-N0248
CAS No.: 58316-41-9
Category:
Umbelliferae/Apiaceae Extract Infection Triterpenes Plant Terpenoids Bupleurum chinensis DC. Extract Disease Research Fields
Target:
2
2 Cited Publications
Cat. No.: HY-P0298A
CAS No.: 23827-91-0
Target:
Research Areas:
2
Category:
Infection Plant Simple Phenylpropanols Phenylpropanoids Other Families Extract Disease Research Fields
Target:
2
2 Cited Publications
Target:
Research Areas:
SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist, with Kis of 0.48 nM and 0.73 nM for B1 kinin receptors of human fibroblast MRC5 and HEK cells expressing human B1 receptors, 481 nM and 358 nM for B2 receptors of guinea pig ileum membranes and CHO cells expressing human B1 receptor, respectively.
2
2 Cited Publications
Cat. No.: HY-P73017
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: EFNB2; Eph-Related Receptor Tyrosine Kinase Ligand 5; Prev. EPLG5; MGC126226; Ephrin-B2; MGC126227; LERK5; MGC126228; HTKL; EPH-Related Receptor Tyrosine Kinase Ligand 5; HTK Ligand; LERK-5; Htk-L; HTK-L; Ephrin B2; Ligand Of Eph-Related Kinase 5
Species:
Mouse
Source:
HEK293
-
-
Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
