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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
2 Results for "
CPI 0610
" in MedChemExpress (MCE) Product Catalog:
Products (2)
2 Results for "CPI 0610" in MCE Product Catalog:
Synonyms: CPI-0610
Target:
Research Areas:
Pelabresib (CPI-0610) is a potent, selective, orally active and cell-active BET inhibitor. Pelabresib inhibits BRD4-BD1 with an IC50 of 39 nM, and with an EC50 value of 0.18 μM for MYC .
Cat. No.: HY-12863B
CAS No.: 1380089-81-5
Research Areas:
CPI-0610 carboxylic acid is a novel small-molecule bromodomain and extraterminal protein inhibitor for the treatment of multiple myeloma. CPI-0610 carboxylic acid binds to the N-terminal bromodomains of BRD2, BRD3, BRD4, and BRDT, as well as the BRD9 bromodomain. CPI-0610 carboxylic acid can serve as a target protein ligand for the synthesis of PROTAC. CPI-0610 carboxylic acid can be used for research on multiple myeloma, acute myeloid leukemia, and lung and cervical cancers .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
