3 Results for "

Monatepil

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "Monatepil" in MCE Product Catalog:

Cat. No.: HY-106818
CAS No.: 103377-41-9
Synonyms: AJ-2615 free base
Monatepil (AJ-2615 free base) is a calcium antagonist with potent α1-adrenoceptor blocking activity. Monatepil inhibits vasopressin- or methacholine-induced ischemic electrocardiographic changes in a rat model of vasospastic angina and reduces the mean arterial pressure in anesthetized rats. Monatepil also enhances low-density lipoprotein (LDL) receptor activity in human skin fibroblasts . Monatepil can be used in research related to hypertension, atherosclerosis, hyperlipidemia and vasospastic angina .
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Cat. No.: HY-106818A
CAS No.: 103379-03-9
Synonyms: AJ-2615
Monatepil (AJ-2615 free base) maleate is a calcium antagonist with potent α1-adrenoceptor blocking activity. Monatepil maleate inhibits vasopressin- or methacholine-induced ischemic electrocardiographic changes in a rat model of vasospastic angina and reduces the mean arterial pressure in anesthetized rats. Monatepil maleate also enhances low-density lipoprotein (LDL) receptor activity in human skin fibroblasts . Monatepil maleate can be used in research related to hypertension, atherosclerosis, hyperlipidemia and vasospastic angina .
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Cat. No.: HY-106818B
CAS No.: 103379-02-8
Synonyms: AJ-2615 hydrochloride
Monatepil (AJ-2615 free base) hydrochloride is a calcium antagonist with potent α1-adrenoceptor blocking activity. Monatepil hydrochloride inhibits vasopressin- or methacholine-induced ischemic electrocardiographic changes in a rat model of vasospastic angina and reduces the mean arterial pressure in anesthetized rats. Monatepil hydrochloride also enhances low-density lipoprotein (LDL) receptor activity in human skin fibroblasts . Monatepil hydrochloride can be used in research related to hypertension, atherosclerosis, hyperlipidemia and vasospastic angina .
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