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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
19 Results for "
Motilin Receptor
" in MedChemExpress (MCE) Product Catalog:
Products (19)
19 Results for "Motilin Receptor" in MCE Product Catalog:
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1 Cited Publications
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DS-3801b is a potent and non-macrolide agonist of GPR38. DS-3801b is expected to be novel gastrointestinal prokinetic agents for the research of functional gastrointestinal disorders such as gastroparesis and chronic constipation .
Cat. No.: HY-P1037
CAS No.: 52906-92-0
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MA-2029 is a selective, orally active, and competitive motilin receptor antagonist (IC50=4.9 nM). MA-2029 is selective for the motilin receptor over various other receptors and ion channels. MA-2029 may be useful for gastrointestinal disorders associated with disturbed gastrointestinal motility .
Cat. No.: HY-P3680
CAS No.: 55524-56-6
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Cat. No.: HY-106327
CAS No.: 110205-60-2
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EM-523 is a motilin agonist and an erythromycin derivative. EM-523 has pED50 values of 8.19 and 6.08 for promoting contractions in rabbit small intestinal tissue and human duodenal tissue, respectively. EM-523 can be used in the research of gastrointestinal diseases .
Cat. No.: HY-105263
CAS No.: 110480-13-2
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EM574 is a potent motilin receptor agonist in the human gastric antrum and rabbit gastrointestinal tract in vitro. EM574 is an erythromycin derivative .
Cat. No.: HY-111232
CAS No.: 874958-63-1
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GSK894281 is an orally active and highly potent ghrelin receptor full agonist with a pEC50 of <4.9 at the human motilin receptor. GSK894281 effectively enters the CNS. GSK894281 has the potential for constipation or to assist in emptying the colon prior to colonoscopy or colon surgery research .
Cat. No.: HY-P1541
CAS No.: 85490-53-5
Synonyms: Motilin (canine)
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Cat. No.: HY-105333
CAS No.: 151052-43-6
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KC-11458 is a motilin agonist. KC-11458 can accelerate gastric emptying .
Cat. No.: HY-171853
CAS No.: 223442-22-6
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RWJ-68022 (Example 9) is a cyclopentene derivative and a motilin receptor antagonist. RWJ-68022 can compete with motilin and erythromycin for the motilin receptor site. RWJ-68022 can be used in the research of gastrointestinal-related diseases .
Cat. No.: HY-106258
CAS No.: 533927-56-9
Synonyms: OHM 11638; BAX-ACC 1638; MOT 288
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Cat. No.: HY-106018
CAS No.: 154738-42-8
Synonyms: GM 611
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Mitemcinal (GM 611) is an oral motilin receptor agonist. Studies in rabbits and dogs have shown that it can promote defecation without causing severe diarrhea, increase stool weight without increasing water content in the rabbit constipation model, and reduce the time to first defecation in dogs. Mitemcinal may be a constipation suppressant due to its early onset and short duration of action .
Cat. No.: HY-106018A
CAS No.: 154802-96-7
Synonyms: GM 611 fumarate
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Mitemcinal fumarate is an oral motilium agonist. Studies in rabbits and dogs have shown that it can promote defecation without causing severe diarrhea, increase stool weight without increasing water content in the rabbit constipation model, and reduce the time to first defecation in dogs. Mitemcinal fumarate may be a constipation suppressant due to its early onset and short duration of action.
Cat. No.: HY-106323
CAS No.: 59530-69-7
Synonyms: KW-5139
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Cat. No.: HY-P1233
CAS No.: 153966-48-4
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Cat. No.: HY-P1233A
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Cat. No.: HY-187989
CAS No.: 33275-72-8
Synonyms: EM-B enol ether
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ME67 (EM-B enol ether) is a motilin receptor (Motilin Receptor) agonist with pIC50 values of 8.38 and 6.49 for rabbit and human motilin receptors, respectively. ME67 activates the G protein-coupled Motilin Receptor, inducing calcium mobilization, calcium flux, receptor internalization, and gastrointestinal motility. ME67 can be used in research on gastrointestinal motility disorders .
Cat. No.: HY-187988
CAS No.: 110469-03-9
Synonyms: N-methyl EM-A
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ME36 (N-methyl EM-A) is a motilin receptor agonist that induces calcium mobilization, with a pIC50 of 7.58 for the rabbit motilin receptor. ME36 can be used in research on digestive system diseases .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
