3 Results for "

Tyr139

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "Tyr139" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-P5963
CAS No.: 2983116-47-6
Target:  

Interleukin Related

Research Areas:  

Inflammation/Immunology

Lib2-1, a macrocyclic peptide, is an IL-17C/IL-17RE interaction inhibitor. Lib2-1 can be used for autoimmune and inflammatory diseases research .
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Cat. No.: HY-189042
CAS No.: 738562-57-7
Target:  

GABA Receptor

Research Areas:  

Neurological Disease

EF1500 is a potent human GABA transporter 1 (hGAT1) inhibitor and a lipophilic THPO analog. EF1500 occupies the binding site by forming a hydrogen bond with active residues of hGAT1 (such as Tyr139) through its exocyclic amino group, thereby blocking GABA reuptake. EF1500 can be used for research on central nervous system diseases .
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Cat. No.: HY-P11623
Research Areas:  

Inflammation/Immunology

4L2-P13D is an IL-11 antagonist with an IC50 of 2.8 μM. 4L2-P13D has a KD of 11 nM for hIL-11. 4L2-P13D exhibits antifibrotic and renoprotective activities. 4L2-P13D can be used in the research of renal fibrosis .
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