3 Results for "

XRP9881

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "XRP9881" in MCE Product Catalog:

Cat. No.: HY-125374
CAS No.: 156294-36-9
Purity:  ≥97.0%
Synonyms: XRP9881
Target:  

Microtubule/Tubulin

Research Areas:  

Neurological Disease Cancer

Larotaxel (XRP9881) is an orally active and blood-brain barrier penetrant Microtubule stabilizer with an IC50 of 0.21 μM. Larotaxel shows activity in Taxane-resistant tumor models. Larotaxel exhibits antitumor activity in intracranial glioblastoma models. Larotaxel can be used for research on advanced solid tumors .
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Cat. No.: HY-125374A
CAS No.: 192573-38-9
Synonyms: XRP9881 dihydrate
Target:  

Microtubule/Tubulin

Larotaxel dihydrate (XRP9881 dihydrate) is an orally active and blood-brain barrier penetrant Microtubule stabilizer with an IC50 of 0.21 μM. Larotaxel dihydrate shows activity in Taxane-resistant tumor models. Larotaxel dihydrate exhibits antitumor activity in intracranial glioblastoma models. Larotaxel dihydrate can be used for research on advanced solid tumors .
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Cat. No.: HY-125374S
Synonyms: XRP9881-d9
Larotaxel-d9 (XRP9881-d9) is the d9-labeled Larotaxel (HY-125374). Larotaxel (XRP9881) is an orally active and blood-brain barrier penetrant Microtubule stabilizer with an IC50 of 0.21 μM. Larotaxel shows activity in Taxane-resistant tumor models. Larotaxel exhibits antitumor activity in intracranial glioblastoma models. Larotaxel can be used for research on advanced solid tumors .
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