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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
1 Result for "
constitutively active mutants
" in MedChemExpress (MCE) Product Catalog:
Products (1)
1 Results for "constitutively active mutants" in MCE Product Catalog:
Cat. No.: HY-W559510A
CAS No.: 746661-90-5
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Research Areas:
MC4R antagonist-3 hydrochloride is a selective melanocortin-4 receptor (MC4R) antagonist with a Kd value of 2 nM. MC4R antagonist-3 hydrochloride binds to MC4R and alters its conformation, specifically promoting ERK1/2 phosphorylation in constitutively active mutants while inhibiting basal cAMP production. MC4R antagonist-3 hydrochloride can be used for research on obesity .
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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
