12 Results for "

5-CT

" in MedChemExpress (MCE) Product Catalog:
Products (12)

12 Results for "5-CT" in MCE Product Catalog:

19
19 Publications Verification
Cat. No.: HY-10985
CAS No.: 437742-34-2
Purity:  99.13%
Synonyms: Salinosporamide A; NPI-0052
Marizomib (Salinosporamide A) is a second-generation, irreversible, brain-penetrant, pan-proteasome inhibitor. Marizomib inhibits the CT-L (β5), CT-T-laspase-like (C-L, β1) and trypsin-like (T-L, β2) activities of the 20S proteasome (IC50=3.5, 28, and 430 nM, respectively) .
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1 Cited Publications
Cat. No.: HY-13527
CAS No.: 192927-92-7
Purity:  98.68%
Target:  

5-HT Receptor

LY310762 is a selective 5-HT1D receptor antagonist with a Ki value of 249 nM for the guinea pig receptor. LY310762 blocks presynaptic 5-HT1D autoreceptors and enhances potassium-stimulated [ 3H]5-HT outflow from guinea pig cortical slices. LY310762 abolishes the inhibitory effect of 5-CT (HY-135555)/L-694,247 (HY-101208) on sympathetic nerve-induced renal vasoconstriction mediated by prejunctional 5-HT1D receptors. LY310762 potentiates the increase in extracellular 5-HT concentration induced by Fluoxetine (HY-B0102). LY310762 is used in research related to depression and diabetic nephropathy .
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Cat. No.: HY-100942
CAS No.: 74885-72-6
Purity:  ≥98.0%
Synonyms: 5-CT maleate
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

5-Carboxamidotryptamine maleate (5-CT maleate) is a potent 5-HT1A, 5-HT1B, 5-HT1D, 5-HT5 and 5-HT7 receptors agonist .
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Cat. No.: HY-135555
CAS No.: 74885-09-9
Purity:  98.74%
Synonyms: 5-CT
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

5-Carboxamidotryptamine (5-CT) is a 5-HT1A, 5-HT1B, 5-HT1D, 5-HT5A, 5-HT7 receptor agonist . 5-Carboxamidotryptamine has a Ki value of 4.6 nM for cloned human 5-HT5A receptor. 5-Carboxamidotryptamine causes a dose-dependent reduction in rectal temperature of mice .
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Cat. No.: HY-100942R
CAS No.: 74885-72-6
Synonyms: 5-CT maleate (Standard)
Research Areas:  

Neurological Disease

5-Carboxamidotryptamine (maleate) (Standard) is the analytical standard of 5-Carboxamidotryptamine (maleate) (HY-100942). This product is intended for research and analytical applications. 5-Carboxamidotryptamine maleate (5-CT maleate) is a potent 5-HT1A, 5-HT1B, 5-HT1D, 5-HT5 and 5-HT7 receptors agonist .
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Cat. No.: HY-124135
CAS No.: 446020-51-5
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

SB-656104 is a potent antagonist of 5-HT7 receptor, with the pKi of 8.70, blocking 5-carboxamidotryptamine (5-CT) stimulated adenylyl cyclase activity .
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Cat. No.: HY-13527A
CAS No.: 379215-96-0
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease Endocrinology

LY310762 free base is a selective 5-HT1D receptor antagonist with a Ki value of 249 nM for the guinea pig receptor. LY310762 free base blocks presynaptic 5-HT1D autoreceptors and enhances potassium-stimulated [ 3H]5-HT outflow from guinea pig cortical slices. LY310762 free base abolishes the inhibitory effect of 5-CT (HY-135555)/L-694,247 (HY-101208) on sympathetic nerve-induced renal vasoconstriction mediated by prejunctional 5-HT1D receptors. LY310762 free base potentiates the increase in extracellular 5-HT concentration induced by Fluoxetine (HY-B0102). LY310762 free base is used in research related to depression and diabetic nephropathy .
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Cat. No.: HY-134483
CAS No.: 851375-22-9
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

5-HT7/5-HT2A receptor antagonist 1 is a high-affinity, orally active, brain-penetrant 5-HT7 and 5-HT2A receptor ligand having a pKi = 8.1 at both receptors. 5-HT7/5-HT2A receptor antagonist 1 behaves as an antagonist in an in vitro functional assay for 5-HT2A and as an inverse agonist in an in vitro functional assay for 5-HT7. 5-HT7/5-HT2A receptor antagonist 1 blockade of 5-Carboxamidotryptamine (5-CT) (HY-135555) induced hypothermia in rats, and blockade of 2,5-dimethoxy-4-iodoamphetamine (DOI) induced head-twitches in mice. 5-HT7/5-HT2A receptor antagonist 1 occupied 5-HT2A receptor binding sites in the frontal cortex of the rat brain. 5-HT7/5-HT2A receptor antagonist 1 can be used for the study of Neurological diseases .
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Cat. No.: HY-P89031
Synonyms: AL5; CT16.3; GAGE-9; GAGEB1; PAGE-1

Host:  

Mouse

Application:  

IHC-P

Reactivity:  

Human

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Cat. No.: HY-P89031A
Synonyms: AL5; CT16.3; GAGE-9; GAGEB1; PAGE-1

Host:  

Mouse

Application:  

IHC-P

Reactivity:  

Human

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Cat. No.: HY-P704517
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: CCN5; ConneCTive Tissue Growth FaCTor-Related Protein 58; Prev. WISP2; WNT1 Inducible Signaling Pathway Protein 2; CTGF-L; CCN Family Member 5; CT58; WNT1-Inducible-Signaling Pathway Protein 2; WISP-2; CTGFL; Cellular Communication Network FaCTor 5; Conne
Species:  
Human
Source:  
E. coli
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